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Recent progress in tetravalent terbium chemistry

D Avignant , E Largeau , Vincent Gaumet , P Dugat , M. El-Ghozzi
Journal of Alloys and Compounds, 1998, 275-277, pp.1-5. ⟨10.1016/S0925-8388(98)00262-X⟩
Journal articles istex hal-02885108v1

(2 R ,3 S )-2-Ammonio-3-hydroxy-3-(4-nitrophenyl)propanoic acid chloride monohydrate

Vincent Gaumet , Valérie Weber , Valery Zaitsev , Michel Madesclaire
Acta Crystallographica Section E : Structure Reports Online [2001-2014], 2008, 64 (6), pp.o1003-o1004. ⟨10.1107/S1600536808012750⟩
Journal articles hal-02885166v1

[(2 R ,3 R )-3-(4-Nitrophenyl)aziridin-2-yl]methanol monohydrate

Vincent Gaumet , C. Denis , F. Leal , M. Madesclaire , V.P. Zaitsev
Acta Crystallographica Section E : Structure Reports Online [2001-2014], 2013, 69 (6), pp.o927-o927. ⟨10.1107/S1600536813013391⟩
Journal articles hal-02885206v1

Development of a freeze-dried kit formulation for the preparation of 99m Tc-NTP 15-5, a radiotracer for scintigraphic imaging of proteoglycans

Aurélien Vidal , Vincent Gaumet , Marie-Josephe Galmier , Sophie Besse , Fernand Leal , et al.
Applied Radiation and Isotopes, 2015, 101, pp.1-9. ⟨10.1016/j.apradiso.2015.03.010⟩
Journal articles hal-01961372v1

Synthesis and biodistribution of technetium-99m-labelled N-(diethylaminoethyl)benzamide via a bis(dithiocarbamate) nitridotechnetium(V) complex

Philippe Auzeloux , Janine Papon , Thierry Masnada , Michèle Borel , Marie-France Moreau , et al.
Journal of Labelled Compounds and Radiopharmaceuticals, 1999, 42 (4), pp.325 - 335. ⟨10.1002/(SICI)1099-1344(199904)42:4<325::AID-JLCR193>3.0.CO;2-J⟩
Journal articles istex hal-01494418v1
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A Novel HPLC Method for Direct Detection of Nitric Oxide Scavengers from Complex Plant Matrices and Its Application to Aloysia triphylla Leaves

Didier Fraisse , Alexandra Degerine-Roussel , Alexis Bred , Samba Ndoye , Magali Vivier , et al.
Molecules, 2018, 23 (7), pp.1574. ⟨10.3390/molecules23071574⟩
Journal articles hal-01873226v1

Mechanism of action of N-phenyl-N′-(2-chloroethyl)ureas in the colchicine-binding site at the interface between α- and β-tubulin

Emmanuel Moreau , Sébastien Fortin , Lianhu Wei , Philippe Labrie , Éric Petitclerc , et al.
Bioorganic and Medicinal Chemistry, 2009, 17 (10), pp.3690 - 3697. ⟨10.1016/j.bmc.2009.03.056⟩
Journal articles hal-01677570v1

A comparative molecular field and comparative molecular similarity indices analyses (CoMFA and CoMSIA) of N-phenyl-N′-(2-chloroethyl)ureas targeting the colchicine-binding site as anticancer agents

Emmanuel Moreau , Sébastien Fortin , Philippe Labrie , Lianhu Wei , Lakshmi P Kotra , et al.
Bioorganic and Medicinal Chemistry, 2008, 16 (4), pp.1914 - 1926. ⟨10.1016/j.bmc.2007.11.004⟩
Journal articles hal-01677579v1

N-Phenyl-N′-(2-chloroethyl)ureas (CEU) as potential antineoplastic agents. Part 2: Role of ω-hydroxyl group in the covalent binding to β-tubulin

Emmanuel Moreau , Sébastien Fortin , Alexandre Patenaude , Michel Desjardins , Jacques Lacroix , et al.
Bioorganic and Medicinal Chemistry, 2007, 15 (3), pp.1430 - 1438. ⟨10.1016/j.bmc.2006.11.005⟩
Journal articles hal-01677583v1

Design, Synthesis, Biological Evaluation, and Structure–Activity Relationships of Substituted Phenyl 4-(2-Oxoimidazolidin-1-yl)benzenesulfonates as New Tubulin Inhibitors Mimicking Combretastatin A-4

Emmanuel Moreau , Sébastien Fortin , Lianhu Wei , Jacques Lacroix , Marie-France Côté , et al.
Journal of Medicinal Chemistry, 2011, 54 (13), pp.4559 - 4580. ⟨10.1021/jm200488a⟩
Journal articles hal-01677554v1

Synthesis, radiofluorination and pharmacological evaluation of a fluoromethyl spirocyclic PET tracer for central σ1 receptors and comparison with fluoroalkyl homologs

Aurélie Maisonial-Besset , Aurélie Maisonial , Eva Grosse Maestrup , Christian Wiese , Achim Hiller , et al.
Bioorganic and Medicinal Chemistry, 2012, 20 (1), pp.257 - 269. ⟨10.1016/j.bmc.2011.11.002⟩
Journal articles istex hal-01677635v1

Radiomarquage du NTP 15-5 ciblant les protéoglycanes pour l’imagerie TEP des pathologies du cartilage : comparaison d’un traceur TEP à un traceur TEMP

C. Valla , V. Gaumet , E. Jouberton , Philippe Auzeloux , F. Degoul , et al.
Médecine Nucléaire - Imagerie Fonctionnelle et Métabolique, 2017, 41 (3), pp.160 - 161. ⟨10.1016/j.mednuc.2017.02.061⟩
Journal articles hal-01677505v1

Synthesis and Biological Evaluation of New Quinoxaline Derivatives of ICF01012 as Melanoma-Targeting Probes

Emmanuel Moreau , Radhia El Aissi , Jianrong Liu , Sophie Besse , Damien Canitrot , et al.
ACS Medicinal Chemistry Letters, 2014, 5 (5), pp.468 - 473. ⟨10.1021/ml400468x⟩
Journal articles hal-01677548v1

Imidazonaphthyridine systems (part 2): Functionalization of the phenyl ring linked to the pyridine pharmacophore and its replacement by a pyridinone ring produces intriguing differences in cytocidal activity

Emmanuel Moreau , Nicolas Masurier , Eric Debiton , Alicia Jacquemet , Antoine Bussière , et al.
European Journal of Medicinal Chemistry, 2012, 52, pp.137 - 150. ⟨10.1016/j.ejmech.2012.03.011⟩
Journal articles istex hal-01677549v1
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A Photochemical Approach to Pyridopyrroloquinoline Derivatives as New Potential Anticancer Agents

Pierre-Jean Aragon , Ange-Désiré Yapi , Frédéric Pinguet , Jean-Michel Chezal , Jean-Claude Teulade , et al.
Chemical and Pharmaceutical Bulletin, 2004, 52, pp.659 - 663. ⟨10.1248/cpb.52.659⟩
Journal articles hal-02384520v1

Antibody functionalization for pretargeted imaging and radiotherapy Nanotechnology for targeted personalized medicines and theranostics

Taiariol Ludivine , Aurélie Rondon , Mercedes Quintana , Sophie Besse , Isabelle Navarro-Teulon , et al.
E-MRS 2018 Spring Meeting, Jun 2018, Strasbourg, France
Conference papers hal-01938907v1
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Base/cryptand/metal-free automated nucleophilic radiofluorination of [ 18 F]FDOPA from iodonium salts: importance of hydrogen carbonate counter ion

Aurélie Maisonial-Besset , Audrey Serre , Ali Ouadi , Sébastien Schmitt , Damien Canitrot , et al.
European Journal of Organic Chemistry, 2018, 2018 (48), pp.7058-7065. ⟨10.1002/ejoc.201801608⟩
Journal articles hal-02343361v1

Reaction of 4-Bromobenzyl-3-methyl-1,2-oxazin-6-ones with Primary Aliphatic Amines. Synthesis and Structural Determination of New Oxazine and Isoxazole Derivatives

Jacques Couquelet , Monique Bebot , Pascal Coudert , Fernand Leal , Jacques Métin , et al.
Heterocycles, 1998, 48 (3), pp.451. ⟨10.3987/COM-97-8050⟩
Journal articles hal-02883844v1

Synthesis and single-crystal structural study of an original low-temperatureform α of BaTbF6

Eric Largeau , Vincent Gaumet , Malika El-Ghozzi , Daniel Avignant , Jean Claude Cousseins
Journal of Materials Chemistry, 1997, 7 (9), pp.1881-1885. ⟨10.1039/A701615H⟩
Journal articles istex hal-02883840v1
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Click and Bioorthogonal Chemistry: The Future of Active Targeting of Nanoparticles for Nanomedicines?

Ludivine Taiariol , Carole Chaix , Carole Farre , Emmanuel Moreau
Chemical Reviews, 2022, 122 (1), pp.340-384. ⟨10.1021/acs.chemrev.1c00484⟩
Journal articles hal-03406814v1
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In vitro cytotoxic effects of secondary metabolites of DEHP and its alternative plasticizers DINCH and DINP on a L929 cell line

Teuta Eljezi , Pierre Pinta , Fabien Nativel , Damien Richard Richard , Jérémy Pinguet , et al.
International Journal of Hygiene and Environmental Health, 2019, 222 (3), pp.583-589. ⟨10.1016/j.ijheh.2019.03.005⟩
Journal articles hal-02385535v1

Design, synthesis and evaluation of targeted hypoxia-activated prodrugs applied to chondrosarcoma chemotherapy

Yvain Gerard , Aurélien Voissière , Caroline Peyrode , Marie-Josephe Galmier , Elise Maubert , et al.
Bioorganic Chemistry, 2020, 98, pp.103747. ⟨10.1016/j.bioorg.2020.103747⟩
Journal articles hal-03437255v1

Linker structure-activity relationships in fluorodeoxyglucose chlorambucil conjugates for tumor-targeted chemotherapy

Valérie Weber , Mostafa El Hilali , Bastien Reux , Eric Debiton , Fernand Leal , et al.
Bioorganic and Medicinal Chemistry, 2017, 25 (20), pp.5692 - 5708. ⟨10.1016/j.bmc.2017.08.043⟩
Journal articles hal-01677115v1

Using the Sonogashira Reaction for Preparing a New Fragment Library based on the 3-alkynylimidazo[1,2-alpha] pyridine Scaffold

Caroline Castera-Ducros , Hussein El-Kashef , Melanie Piednoel , Vincent Remusat , Jean-Claude Teulade , et al.
Letters in Organic Chemistry, 2016, 13 (7), pp.519-525. ⟨10.2174/1570178613666160919124456⟩
Journal articles hal-01460673v1

Characterization of the Covalent Binding of N-Phenyl-N'-(2-chloroethyl)ureas to -Tubulin: Importance of Glu198 in Microtubule Stability

Emmanuel Moreau , S. Fortin , B. Bouchon , C. Chambon , J. Lacroix , et al.
Journal of Pharmacology and Experimental Therapeutics, 2011, 336 (2), pp.460 - 467. ⟨10.1124/jpet.110.171082⟩
Journal articles hal-01677562v1

Radiosynthesis and Radiotracer Properties of a 7-(2-[18F]Fluoroethoxy)-6-methoxypyrrolidinylquinazoline for Imaging of Phosphodiesterase 10A with PET

Aurélie Maisonial-Besset , Uta Funke , Winnie Deuther-Conrad , Gregor Schwan , Aurélie Maisonial , et al.
Pharmaceuticals Policy and Law, 2012, 5 (12), pp.169 - 188. ⟨10.3390/ph5020169⟩
Journal articles hal-01677646v1

N-Substituted 4-aminobenzamides (procainamide analogs): an assessment of multiple cellular effects vis-a-vis ion trapping

Emmanuel Moreau , G. Morissette
Molecular Pharmacology, 2008, ⟨10.1124/mol.105.016527⟩
Journal articles hal-01677587v1

Optimized N-phenyl-N′-(2-chloroethyl)ureas as potential antineoplastic agents: Synthesis and growth inhibition activity

Emmanuel Moreau , Sébastien Fortin , Michel Desjardins , Jean L C Rousseau , Eric Petitclerc , et al.
Bioorganic and Medicinal Chemistry, 2005, 13 (24), pp.6703 - 6712. ⟨10.1016/j.bmc.2005.07.048⟩
Journal articles hal-01677590v1

Heterocyclization of Functionalized Vinylic Derivatives of Imidazo[1,2- a ]pyridines

Emmanuel Moreau , Jean Chezal , Gregory Delmas , Alain Gueiffier , Yves Blache , et al.
Journal of Organic Chemistry, 2001, 66 (20), pp.6576 - 6584. ⟨10.1021/jo015582x⟩
Journal articles istex hal-01677665v1
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Inter-individual variability of protein patterns in saliva of healthy adults

Mercedes Quintana , Mercédès Quintana , Olivier Palicki , Géraldine Lucchi , Patrick Ducoroy , et al.
Journal of Proteomics, 2009, 72 (5), pp.822-830. ⟨10.1016/j.jprot.2009.05.004⟩
Journal articles hal-02454652v1